簡(jiǎn)要描述:英文名稱(chēng): ALK-5 Inhibitor產(chǎn)品應用: TGF-β信號通路調控中國俗稱(chēng): ALK-5 抑制劑 注冊品牌: StemRD 生產(chǎn)廠(chǎng)家: 美國StemRD公司訂購貨號: ALK-50規格型號: 50mg保存溫度: ﹣20℃產(chǎn)品種類(lèi): 小分子工具到貨時(shí)間: 1~5天
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產(chǎn)品英文名稱(chēng):ALK-5 Inhibitor
產(chǎn)品中文名稱(chēng):ALK-5 抑制劑
ALK-5 產(chǎn)品英文簡(jiǎn)述:
A selective inhibitor of ALK5 (TGF-beta type I receptor). It has also been shown that this compound can replace Sox2 when reprogramming cells to iPS cells. 2-(3-(6-METHYLPYRIDIN-2-YL)-1H-PYRAZOL-4-YL)-1,5-NAPHTHYRIDINE
Ref: Gellibert, F., et al. (2004) Identification of 1, 5-naphthyridine derivatives as a novel series of potent and selective TGF-beta type I receptor inhibitors. J Med Chem 47: 4494-4506. Ichida, J.K., et al. (2009) A small-molecule inhibitor of Tgf-beta signaling replaces Sox2 in reprogramming by inducing Nanog. Cell Stem Cell 5: 491-503
Purity: Greater than 98% as determined by LC/MS analysis. LC/MS and/or NMR data available upon request.
Biological Activity :Not determined.
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