簡(jiǎn)要描述:英文名稱(chēng): A83-01產(chǎn)品應用: TGF-β信號通路調控中國俗稱(chēng): TGF-β受體抑制劑 注冊品牌: StemRD 生產(chǎn)廠(chǎng)家: 美國StemRD公司訂購貨號: A8-50規格型號: 50mg保存溫度: ﹣20℃產(chǎn)品種類(lèi): 小分子工具到貨時(shí)間: 1~5天
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產(chǎn)品英文名稱(chēng):A83-01
產(chǎn)品中文名稱(chēng):A83-01
訂購:
A83-01 產(chǎn)品英文簡(jiǎn)述:
A selective inhibitor of ALK-4 (Activin/Nodal receptor), ALK-5 (TGF-β type I receptor), and ALK-7 (nodal receptor). Only weakly inhibits ALK-1, -2, -3, and -6. 3-(6-METHYLPYRIDIN-2-YL)-1-PHENYLTHIOCARBAMOYL-4-QUINOLIN-4-YLPYRAZOLE
Ref: Tojo, M., et al. The ALK-5 inhibitor A-83-01 inhibits Smad signaling and epithelial-to-mesenchymal transition by transforming growth factor-beta. Cancer Sci. 96: 791-800, 2005.
Purity: Greater than 98% as determined by LC/MS analysis. LC/MS and/or NMR data available upon request.
Biological Activity: Not determined.
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