簡(jiǎn)要描述:英文名稱(chēng): CHIR99021產(chǎn)品應用: WNT信號通路調控中國俗稱(chēng): CHIR99021 注冊品牌: StemRD 生產(chǎn)廠(chǎng)家: 美國StemRD公司訂購貨號: CHIR-10規格型號: 10mg保存溫度: ﹣20℃產(chǎn)品種類(lèi): 小分子工具到貨時(shí)間: 1~5天
產(chǎn)品目錄
相關(guān)文章
產(chǎn)品英文名稱(chēng): CHIR99021
產(chǎn)品中文名稱(chēng): CHIR99021
訂購:
CHIR99021產(chǎn)品英文簡(jiǎn)述:
CHIR99021 (CT99021) is a glycogen synthase kinase 3β (GSK3β) inhibitor with IC50 less than 10 nM. Compared to other GSK-3 inhibitors, CHIR-99201 does not exhibit cross-reactivity against cyclin-dependent kinases (CDKs) with 350-fold selectivity toward GSK-3β compared to CDKs .
Ref: Tighe A et al. BMC Cell Biol. 2007 Aug 14;8:34
Purity: Greater than 99% as determined by LC/MS analysis. LC/MS and/or NMR data available upon request.
Biological Activity: In a cell-based assay measuring the activation of the TCF reporter gene, this compound gives EC50 of 50 nM.
如果想了解更多華雅干技術(shù)有限公司在中國代理銷(xiāo)售系列產(chǎn)品,咨詢(xún)與購買(mǎi)!
:勾娜娜
:
:
電話(huà)
微信掃一掃